黄体制剂（英语：Progestin）是一种合成的[1]孕激素，与孕酮有类似效果。[2]Progestin的两种最重要用途为激素避孕（独立或与雌激素一同使用）以及作为激素替代疗法预防不受对抗的雌激素导致的子宫内膜增生。
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| | 雌激素 | ER（雌激素受体）
激动剂 |
- （甾体类） Alfatradiol
- 某些雄激素/合成类固醇(e.g., testosterone, testosterone esters, methyltestosterone, metandienone, nandrolone esters) (via estrogenic metabolites)
- 某些黄体制剂 (例如：诺瑞酮，左炔诺孕酮二醋酸酯，替前列酮)
- 氯米酮
- 醋酸邻雌二醇
- 共轭雌三醇
- 共轭雌激素
- 环雌三醇
- 环雌甲酮
- 酯化雌激素
- 雌四醇†
- 雌二醇
- Estradiol esters (e.g., estradiol acetate, estradiol benzoate, estradiol cypionate, estradiol enanthate, estradiol undecylate, estradiol valerate, polyestradiol phosphate, estradiol ester mixtures (Climacteron))
- Estramustine phosphate
- Estriol
- Estriol esters (e.g., estriol succinate, polyestriol phosphate)
- Estrogenic substances
- Estrone
- Estrone esters
- * Estrone sulfate
- * Estropipate (piperazine estrone sulfate)
- Ethinylestradiol#
- * Ethinylestradiol sulfonate
- Hydroxyestrone diacetate
- Mestranol
- Methylestradiol
- Moxestrol
- Nilestriol
- Prasterone (dehydroepiandrosterone; DHEA)
- Prasterone enanthate
- Prasterone sulfate
- Promestriene
- Quinestradol
- Quinestrol
- （非甾体类） Benzestrol
- Bifluranol
- Chlorotrianisene
- Dienestrol
- 双乙酸双烯雌酚
- 乙烯雌酚（己烯雌酚(stilbestrol)）
- Diethylstilbestrol esters/ethers
- Dimestrol (diethylstilbestrol dimethyl ether)
- Fosfestrol (diethylstilbestrol diphosphate)
- Mestilbol (diethylstilbestrol monomethyl ether)
- Doisynoestrol (fenocycline)
- Hexestrol
- Hexestrol esters
- Methallenestril
- Methestrol (promethestrol)
- Methestrol dipropionate (promethestrol dipropionate)
- Paroxypropione
- Quadrosilan
- Triphenylbromoethylene
- Triphenylchloroethylene
- Zeranol
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| | 促性腺激素 | |
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| | 抗雌激素 | ER拮抗剂
(包含SERMs/SERDs) | |
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| | 芳香酶抑制剂 | |
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| | 抗性腺激素 |
- 雄激素/合成类固酮 (例如 睾酮, 睾酮酯, nandrolone esters, oxandrolone, 氟氧孕酮)
- D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride)
- GnRH agonists (e.g., leuprorelin, goserelin)
- GnRH antagonists (e.g., cetrorelix, elagolix)
- Progestogens (e.g., chlormadinone acetate, cyproterone acetate, gestonorone caproate, hydroxyprogesterone caproate, medroxyprogesterone acetate, megestrol acetate)
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| | 其他 | |
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