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再摄取强化剂:修订间差异

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一些再攝取增強劑:
一些再攝取增強劑:


{{tsl|en|Coluracetam||Coluracetam}}是一種膽鹼再攝取強化劑<ref name="PMID18461272">[http://www.ncbi.nlm.nih.gov/pubmed/18461272 MKC-231, a choline-uptake enhancer: long-lasting cognitive improvement after repeated administration in AF64A-treated rats.], Pubmed.</ref>。[[黄酮类]][[木犀草素]]以及它的一些[[衍生物]]可增強[[多巴胺轉運體]]的再攝取作用<ref name="pmid19815045">{{cite journal |vauthors=Zhao G, Qin GW, Wang J, Chu WJ, Guo LH |title=Functional activation of monoamine transporters by luteolin and apigenin isolated from the fruit of Perilla frutescens (L.) Britt |journal=Neurochem. Int. |volume=56 |issue=1 |pages=168–76 |year=2010 |pmid=19815045 |doi=10.1016/j.neuint.2009.09.015 |url=}}</ref><ref name="pmid20971650">{{cite journal |vauthors=Zhang J, Liu X, Lei X, etal |title=Discovery and synthesis of novel luteolin derivatives as DAT agonists |journal=Bioorg. Med. Chem. |volume=18 |issue=22 |pages=7842–8 |year=2010 |pmid=20971650 |doi=10.1016/j.bmc.2010.09.049 |url=}}</ref>。''Caulis Sinomenii'' 的萃取物可增加[[多巴胺|DA]]/[[正腎上腺素|NE]]的再攝取<ref name="pmid19491370">{{cite journal |vauthors=Zhao G, Bi C, Qin GW, Guo LH |title=Caulis Sinomenii extracts activate DA/NE transporter and inhibit 5HT transporter |journal=Exp. Biol. Med. (Maywood) |volume=234 |issue=8 |pages=976–85 |year=2009 |pmid=19491370 |doi=10.3181/0903-RM-92 |url=}}</ref>。
{{tsl|en|Coluracetam||Coluracetam}}是一種膽鹼再攝取強化劑<ref name="PMID18461272">[http://www.ncbi.nlm.nih.gov/pubmed/18461272 MKC-231, a choline-uptake enhancer: long-lasting cognitive improvement after repeated administration in AF64A-treated rats.] {{Wayback|url=http://www.ncbi.nlm.nih.gov/pubmed/18461272 |date=20190904014740 }}, Pubmed.</ref>。[[黄酮类]][[木犀草素]]以及它的一些[[衍生物]]可增強[[多巴胺轉運體]]的再攝取作用<ref name="pmid19815045">{{cite journal |vauthors=Zhao G, Qin GW, Wang J, Chu WJ, Guo LH |title=Functional activation of monoamine transporters by luteolin and apigenin isolated from the fruit of Perilla frutescens (L.) Britt |journal=Neurochem. Int. |volume=56 |issue=1 |pages=168–76 |year=2010 |pmid=19815045 |doi=10.1016/j.neuint.2009.09.015 |url=}}</ref><ref name="pmid20971650">{{cite journal |vauthors=Zhang J, Liu X, Lei X, etal |title=Discovery and synthesis of novel luteolin derivatives as DAT agonists |journal=Bioorg. Med. Chem. |volume=18 |issue=22 |pages=7842–8 |year=2010 |pmid=20971650 |doi=10.1016/j.bmc.2010.09.049 |url=}}</ref>。''Caulis Sinomenii'' 的萃取物可增加[[多巴胺|DA]]/[[正腎上腺素|NE]]的再攝取<ref name="pmid19491370">{{cite journal |vauthors=Zhao G, Bi C, Qin GW, Guo LH |title=Caulis Sinomenii extracts activate DA/NE transporter and inhibit 5HT transporter |journal=Exp. Biol. Med. (Maywood) |volume=234 |issue=8 |pages=976–85 |year=2009 |pmid=19491370 |doi=10.3181/0903-RM-92 |url=}}</ref>。


==参见==
==参见==

2020年12月20日 (日) 14:19的版本

Coluracetam英语Coluracetam,一種高親和力膽鹼攝取(HACU)增強劑。

再攝取強化劑 (Reuptake Enhancer , RE),有時也稱作再攝取激活劑,是一種再攝取調節劑。可以增強膜上轉運蛋白神經遞質再攝取,使胞外神經遞質浓度下降,進而導致較少的神經傳導英语neurotransmission

一些再攝取增強劑:

Coluracetam英语Coluracetam是一種膽鹼再攝取強化劑[1]黄酮类木犀草素以及它的一些衍生物可增強多巴胺轉運體的再攝取作用[2][3]Caulis Sinomenii 的萃取物可增加DA/NE的再攝取[4]

参见

参考资料

  1. ^ MKC-231, a choline-uptake enhancer: long-lasting cognitive improvement after repeated administration in AF64A-treated rats.页面存档备份,存于互联网档案馆), Pubmed.
  2. ^ Zhao G, Qin GW, Wang J, Chu WJ, Guo LH. Functional activation of monoamine transporters by luteolin and apigenin isolated from the fruit of Perilla frutescens (L.) Britt. Neurochem. Int. 2010, 56 (1): 168–76. PMID 19815045. doi:10.1016/j.neuint.2009.09.015. 
  3. ^ Zhang J, Liu X, Lei X, et al. Discovery and synthesis of novel luteolin derivatives as DAT agonists. Bioorg. Med. Chem. 2010, 18 (22): 7842–8. PMID 20971650. doi:10.1016/j.bmc.2010.09.049. 
  4. ^ Zhao G, Bi C, Qin GW, Guo LH. Caulis Sinomenii extracts activate DA/NE transporter and inhibit 5HT transporter. Exp. Biol. Med. (Maywood). 2009, 234 (8): 976–85. PMID 19491370. doi:10.3181/0903-RM-92.